The small-molecule 3G11 inhibits HIV-1 reverse transcription
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چکیده
منابع مشابه
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Members of the ETS transcription factor family have been implicated in several cancers,where they are often dysregulated by genomic derangement. ETS variant 1 (ETV1) is an ETS factor gene that undergoes chromosomal translocation in prostate cancers and Ewing sarcomas, amplification in melanomas, and lineage dysregulation in gastrointestinal stromal tumors. Pharmacologic perturbation of ETV1 wou...
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Affiliations: 1 Dana Farber Cancer Institute, Boston, MA, USA 2 Broad Institute, Cambridge, MA, USA 3 Novartis Institute for Biomedical Research, Cambridge, MA, USA 4 Department of Biological Engineering, MIT, Cambridge, MA, USA 5 Koch Institute for Integrative Cancer Research, MIT, Cambridge, MA, USA # Current address: Blueprint medicines, Cambridge, MA, USA *Corresponding author: Levi A Garra...
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ژورنال
عنوان ژورنال: Chemical Biology & Drug Design
سال: 2016
ISSN: 1747-0277
DOI: 10.1111/cbdd.12886